About 9 results found for searched term "5-HT2C agonist-3" (0.121 seconds)
Cat.No. | Name | Target |
---|---|---|
M41740 | 5-HT2C agonist-3 free base | 5-HT Receptor |
5-HT2C agonist-3 ((+)-19) free base is a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM). | ||
M41743 | 5-HT2C agonist-3 | 5-HT Receptor |
5-HT2C agonist-3 ((+)-19) is a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM). | ||
M8864 | Zotepine | 5-HT Receptor |
Zotepine is a potent 5-HT2A, 5-HT2C, histamine H1, α1-adrenergic, and dopamine D2 receptor antagonist with Kd values of 2.6 nM, 3.2 nM, 3.3 nM, 7.3 nM, and 8 nM, respectively. | ||
M30773 | SCH-23390 maleate | Dopamine Receptor |
R-(+)-SCH-23390 maleate | ||
SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively. SCH-23390 maleate is a potent and high efficacy human 5-HT2C receptor agonist with a Ki of 9.3 nM. SCH-23390 maleate also binds with high affinity to the 5-HT2 and 5-HT1C receptors. SCH-23390 maleate inhibits G protein-coupled inwardly rectifying potassium (GIRK) channels with an IC50 of 268 nM. | ||
M41735 | 5-HT2 agonist-1 free base | 5-HT Receptor |
5-HT2 agonist-1 free base is a 5-HT2A & 5-HT2B & 5-HT2C agonist, with IC50s of 10 nM, 8.3, and 1.6 nM respectively. | ||
M41738 | 5-HT2 agonist-1 | 5-HT Receptor |
5-HT2 agonist-1 is a 5-HT2A & 5-HT2B & 5-HT2C agonist, with IC50s of 10 nM, 8.3, and 1.6 nM respectively. | ||
M56097 | SB 243213 | 5-HT Receptor |
SB 243213 is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. | ||
M56084 | SB 243213 hydrochloride | 5-HT Receptor |
SB 243213 hydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. | ||
M56078 | SB 243213 dihydrochloride | 5-HT Receptor |
SB 243213 dihydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. |
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