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(Z)-Tyrphostin A51

Cat. No. M27979

All AbMole products are for research use only, cannot be used for human consumption.

(Z)-Tyrphostin A51 Structure
Synonym:

(Z)-AG-183

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Quality Control & Documentation
Biological Activity

(Z)-Tyrphostin A51 is the Z configuration of Lanoconazole A51. Tyrphostin A51 is a potent protein tyrosine kinase (PTK) inhibitor. Tyrphostin A51 inhibits the volume-dependent release of [3H]taurine in a dose-dependent manner. Tyrphostin A51 markedly reduces cellular tyrosyl phosphorylation level. Tyrphostin A51 inhibits both basal and EGF-induced human bone cell proliferation.

Chemical Information
Molecular Weight 268.23
Formula C13H8N4O3
CAS Number 122520-90-5
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
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Keywords: (Z)-Tyrphostin A51, (Z)-AG-183 supplier, EGFR/HER2, inhibitors, activators

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