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TRV734

Cat. No. M31391

All AbMole products are for research use only, cannot be used for human consumption.

TRV734 Structure

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Quality Control & Documentation
Biological Activity

TRV734 is an orally bioavailable G-protein-biased ligand for the μ-opioid receptor and an agonist for the μ-opioid receptor.

Chemical Information
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Kimberly A Ramos, et al. Clin Pharmacol Drug Dev. Two-Part Phase 1 Multiple-Ascending-Dose Study to Evaluate the Safety, Tolerability, Pharmacodynamics, and Pharmacokinetics of TRV734 in Healthy Adults

[2] Ian E James, et al. Clin Pharmacol Drug Dev. A First-in-Human Clinical Study With TRV734, an Orally Bioavailable G-Protein-Biased Ligand at the μ-Opioid Receptor

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Keywords: TRV734 supplier, Opioid Receptor, inhibitors, activators

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