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TC LPA5 4 is a specific non-lipid LPA5 (GPR92) antagonist (IC50=0.8 μM in LPA5-RH7777 cells). Shows selectivity for LPA5 against 80 other screening targets.TC LPA5 4 was shown to inhibit LPA-induced aggregation of isolated human platelets.TC LPA5 4 inhibits proliferation and migration of thyroid cancer cells.
| Molecular Weight | 410.89 |
| Formula | C23H23ClN2O3 |
| CAS Number | 1393814-38-4 |
| Solubility (25°C) | DMSO ≥ 60 mg/mL |
| Storage | 2-8℃, protect from light, dry, sealed |
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