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SJ6986

Cat. No. M21152

All AbMole products are for research use only, cannot be used for human consumption.

SJ6986  Structure
Size Price Availability Quantity
1mg USD 30  USD30 In stock
5mg USD 60  USD60 In stock
10mg USD 95  USD95 In stock
25mg USD 185  USD185 In stock
50mg USD 300  USD300 In stock
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Quality Control & Documentation
Biological Activity

SJ6986 is a potent, selective, and orally effective GSPT1/2 degradation agent with a DC50 value of 2.1 nM (Dmax 99%) for GSPT1.

Chemical Information
Molecular Weight 497.40
Formula C20H14F3N3O7S
CAS Number 2765625-93-0
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Gisele Nishiguchi, et al. J Med Chem. Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators

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Keywords: SJ6986 supplier, inhibitors, activators

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