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Ranolazine (CVT 303) is an anti-angina and anti-ischemia agent that works by inhibiting the late effects of inward sodium current (IC50 values of 6 μM and 12 μM for INa and IKr, respectively) without affecting heart rate or blood pressure. Ranolazine is also a partial inhibitor of fatty acid oxidation (FAO).
| Molecular Weight | 500.46 |
| Formula | C24H35Cl2N3O4 |
| CAS Number | 95635-56-6 |
| Form | Solid |
| Solubility (25°C) | DMSO 100mg/ml water 100mg/ml |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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