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Radotinib

Cat. No. M5916

All AbMole products are for research use only, cannot be used for human consumption.

Radotinib Structure
Synonym:

IY-5511

Size Price Availability Quantity
5mg USD 50  USD50 In stock
10mg USD 75  USD75 In stock
25mg USD 140  USD140 In stock
50mg USD 240  USD240 In stock
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Quality Control & Documentation
Biological Activity

Radotinib is a selective BCR-ABL1 tyrosine kinase inhibitor with IC50 of 34 nM, used to treat Chronic Myeloid Leukemia.

Chemical Information
Molecular Weight 530.50
Formula C27H21F3N8O
CAS Number 926037-48-1
Solubility (25°C) 100 mg/mL in DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Kim SH, et al. Haematologica. Efficacy and safety of radotinib in chronic phase chronic myeloid leukemia patients with resistance or intolerance to BCR-ABL1 tyrosine kinase inhibitors.

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Keywords: Radotinib, IY-5511 supplier, Src-bcr-Abl, inhibitors, activators

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