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OPC 21268

Cat. No. M7084

All AbMole products are for research use only, cannot be used for human consumption.

OPC 21268 Structure
Synonym:

Fuscoside

Size Price Availability Quantity
1mg USD 50  USD50 In stock
5mg USD 95  USD95 In stock
10mg USD 130  USD130 In stock
25mg USD 210  USD210 In stock
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Quality Control & Documentation
Biological Activity

OPC 21268 is a nonpeptide vasopressin V1 receptor antagonist. Displays greater affinity for rat V1 than human V1 (Ki values are 25 and 8800 nM respectively). Exhibits 1000-fold selectivity for V1 receptors over V2 receptors. Orally active.

Chemical Information
Molecular Weight 449.54
Formula C26H31N3O4
CAS Number 131631-89-5
Solubility (25°C) DMSO 44.95 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Chan, et al. Cell. Pharmacological inactivation of Skp2 SCF ubiquitin ligase restricts cancer stem cell traits and cancer progression.

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Keywords: OPC 21268, Fuscoside supplier, inhibitors, activators

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