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NVS-PAK1-C is a potent, ATP-competitive and specific allosteric PAK1 inhibitor probe with IC50 values of 5 nM and 6 nM for dephosphorylated PAK1 and phosphorylated PAK1, respectively. NVS-PAK1-C is also against dephosphorylated PAK2 (IC50=270 nM) and phosphorylated PAK2 (IC50=720 nM).
| Molecular Weight | 465.9 |
| Formula | C22H23ClF3N5O |
| CAS Number | 2250019-95-3 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Related PAK Products |
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| PF-3758309 dihydrochloride
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