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LDC1267

Cat. No. M11231

All AbMole products are for research use only, cannot be used for human consumption.

LDC1267  Structure
Size Price Availability Quantity
5mg USD 78  USD78 In stock
10mg USD 127  USD127 In stock
25mg USD 225  USD225 In stock
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Quality Control & Documentation
Biological Activity

LDC1267 is a highly selective inhibitor of TAM (Tyro3,Axl and Mer) kinases with IC50 values of <5 nM/8 nM/29 nM against Tyro3/Axl/Mer, respectively.

Chemical Information
Molecular Weight 560.55
Formula C30H26F2N4O5
CAS Number 1361030-48-9
Form Solid
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Daria Zdżalik-Bielecka, et al. Mol Cancer Res. Bemcentinib and Gilteritinib Inhibit Cell Growth and Impair the Endo-Lysosomal and Autophagy Systems in an AXL-Independent Manner

[2] Zaofeng Zou, et al. Evid Based Complement Alternat Med. Tyrosine Kinase Receptors Axl and MerTK Mediate the Beneficial Effect of Electroacupuncture in a Cuprizone-Induced Demyelinating Model

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DS-1205b free base 

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Ningetinib Tosylate

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  Catalog
Abmole Inhibitor Catalog




Keywords: LDC1267 supplier, TAM Receptor, inhibitors, activators

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