Free shipping on all orders over $ 500

HSK16149

Cat. No. M21118

All AbMole products are for research use only, cannot be used for human consumption.

HSK16149  Structure

Price and Availability

For this product's availability, delivery time and price, please email [email protected] directly or click the "Inquiry Now" button below.


Quality Control & Documentation
Biological Activity

HSK16149 is an oral γ-aminobutyric acid analog and a novel voltage-gated calcium channel (VGCC) α2δ subunit ligand for studies related to diabetic peripheral neuralgia (DPNP).

Chemical Information
Molecular Weight 209.28
Formula C12H19NO2
CAS Number 2209104-84-5
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Xiaoli Gou, et al. J Pharmacol Exp Ther. Pharmacology and Mechanism of Action of HSK16149, a Selective Ligand of α 2 δ Subunit of Voltage-Gated Calcium Channel with Analgesic Activity in Animal Models of Chronic Pain

Related Calcium Channel Products
CBD3063

CBD3063 is a selective, first-in-class, CRMP2-based peptidomimetic small molecule, which allosterically regulates Cav2.2 to achieve analgesia and pain relief without negative side effect profiles.

TTA-A8 

TTA-A8 is a short-acting T-type calcium channel antagonist with oral activity, exhibiting an IC50 value of 31.3 nM in the FLIPR depolarization assay.

MONIRO-1 

MONIRO-1 is a T-type and N-type calcium channel blocker with IC50 values of 34, 3.3, 1.7 and 7.2 µM against hCav2.2, hCav3.1, hCav3.2 and hCav3.3, respectively.

Azumolene

Azumolene (EU4093 free base), a Dantrolene analog, is a muscle relaxant.

Nexopamil 

Nexopamil is a calcium antagonist of Ca2+ channel, 5HT2, 5HT1A, 5HT1C and dopamine D2 receptors.

  Catalog
Abmole Inhibitor Catalog




Keywords: HSK16149 supplier, Calcium Channel, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.