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GSK251 

Cat. No. M29271

All AbMole products are for research use only, cannot be used for human consumption.

GSK251  Structure

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Quality Control & Documentation
Biological Activity

GSK251 is a highly potent, highly selective, orally bioavailable inhibitor of PI3Kδ with a novel binding mode.

Chemical Information
Molecular Weight 584.71
Formula C29H37FN6O4S
CAS Number 2125968-05-8
Form Solid
Solubility (25°C) DMSO 62.5 mg/mL (ultrasonic and warming and heat to 60°C)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Kenneth Down, et al. J Med Chem. Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode

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  Catalog
Abmole Inhibitor Catalog




Keywords: GSK251  supplier, PI3K, inhibitors, activators

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