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GSK1521498 is a potent and selective μ-opioid receptor antagonist. GSK1521498 dose-dependently reduced both cue-controlled alcohol seeking and alcohol intake in the instrumental context as well as alcohol intake in the choice procedure.
Molecular Weight | 402.44 |
Formula | C24H20F2N4 |
CAS Number | 1007573-18-3 |
Solubility (25°C) | DMSO ≥ 6 mg/mL |
Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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