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GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
| Molecular Weight | 394.47 |
| Formula | C22H26N4O3 |
| CAS Number | 901245-65-6 |
| Solubility (25°C) | DMSO 6 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Goutham Atla, et al. Genome Biol. Genetic regulation of RNA splicing in human pancreatic islets
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