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GSK 4716

Cat. No. M6165

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GSK 4716 Structure
Size Price Availability Quantity
5mg USD 50  USD50 In stock
10mg USD 75  USD75 In stock
50mg USD 320  USD320 In stock
100mg USD 565  USD565 In stock
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Quality Control & Documentation
Biological Activity

GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.

Chemical Information
Molecular Weight 282.33
Formula C17H18N2O2
CAS Number 101574-65-6
Solubility (25°C) 10 mM in DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Saili KS, et al. Toxicology. Neurodevelopmental low-dose bisphenol A exposure leads to early life-stage hyperactivity and learning deficits in adult zebrafish.

[2] Kim Y, et al. J Comb Chem. Efficient discovery of selective small molecule agonists of estrogen-related receptor gamma using combinatorial approach.

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Keywords: GSK 4716 supplier, Estrogen Receptor, inhibitors, activators

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