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GR 89696 fumarate

Cat. No. M6765

All AbMole products are for research use only, cannot be used for human consumption.

GR 89696 fumarate Structure

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Quality Control & Documentation
Biological Activity

GR 89696 fumarate is a highly potent and selective κ-opioid agonist (IC50 = 0.04 nM) that may be selective for the putative κ2 receptor. Anti-nociceptive and neuroprotective in vivo.

Chemical Information
Molecular Weight 530.4
Formula C19H25Cl2N3O3.C4H4O4
CAS Number 126766-32-3
Solubility (25°C) Water 13.26 mg/mL (with gentle warming)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Lanvin, et al. J Biol Chem. Potentiation of ICI182,780 (Fulvestrant)-induced estrogen receptor-alpha degradation by the estrogen receptor-related receptor-α inverse agonist XCT790.

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