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EZH2-IN-4 is an orally active, potent EZH2 inhibitor with IC50s of 0.923 nM and 2.65 nM against wild type (WT) 5-membered (5-mer) EZH2 and mutant 5-mer EZH2, respectively. EZH2-IN-4 has anti-cancer activity.
| Molecular Weight | 511.72 |
| Formula | C29H41N3O3S |
| CAS Number | 2088132-99-2 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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Products are for research use only. Not for human use. We do not sell to patients.
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