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Evatanepag

Cat. No. M10679

All AbMole products are for research use only, cannot be used for human consumption.

Evatanepag Structure
Synonym:

CP-533536 free acid

Size Price Availability Quantity
5mg USD 238  USD238 In stock
10mg USD 365  USD365 In stock
25mg USD 740  USD740 In stock
50mg USD 1150  USD1150 In stock
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Quality Control & Documentation
Biological Activity

Evatanepag (CP-533536 free acid) is a potent selective EP2 receptor agonist with an IC50 of 50 nM for rEP2.

Chemical Information
Molecular Weight 468.57
Formula C25H28N2O5S
CAS Number 223488-57-1
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage -20°C protect from light dry
References

[1] Changxiu Qu, et al. Sci Adv. Ligand recognition, unconventional activation, and G protein coupling of the prostaglandin E 2 receptor EP2 subtype

[2] Claire Veryard. IDrugs. American Society for Clinical Pharmacology and Therapeutics (ASCPT)-111th annual meeting. 17-20 March 2010, Atlanta, GA, USA

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Keywords: Evatanepag, CP-533536 free acid supplier, Prostaglandin Receptor, inhibitors, activators

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