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CPUY074020 

Cat. No. M30844

All AbMole products are for research use only, cannot be used for human consumption.

CPUY074020  Structure

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Quality Control & Documentation
Biological Activity

CPUY074020 is a potent and oral bioavailable inhibitor of histone methyltransferase G9a, with an IC50 of 2.18 μM. CPUY074020 possesses anti-proliferative activity.

Chemical Information
Molecular Weight 416.52
Formula C25H28N4O2
CAS Number 902279-44-1
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Wei-Lin Chen, et al. Bioorg Med Chem. Discovery, design and synthesis of 6H-anthra[1,9-cd]isoxazol-6-one scaffold as G9a inhibitor through a combination of shape-based virtual screening and structure-based molecular modification

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  Catalog
Abmole Inhibitor Catalog




Keywords: CPUY074020  supplier, Histone Methyltransferase, inhibitors, activators

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