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C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and increases the binding between β-catenin and p300. C-82 inhibits the activation of isolated primary mouse quiescent hepatic stellate cells (HSCs) and promotes cell death in culture-activated HSCs.
| Molecular Weight | 578.66 |
| Formula | C33H34N6O4 |
| CAS Number | 1422253-37-9 |
| Solubility (25°C) | DMSO ≥ 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Kangkang Zhang, et al. Nat Nanotechnol. A Gd@C82 single-molecule electret
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