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BMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. BMS-986020 sodium inhibits bile acid and phospholipid transporters with IC50s of 4.8 µM, 6.2 µM, and 7.5 µM for BSEP, MRP4, and MDR3, respectively. BMS-986020 sodium has the potential for the treatment of idiopathic pulmonary fibrosis (IPF).
| Molecular Weight | 504.51 |
| CAS Number | 1380650-53-2 |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage | 2-8°C, dry, sealed |
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