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β-Casomorphin, human TFA

Cat. No. M21325
β-Casomorphin, human TFA Structure
Synonym:

Human β-casomorphin 7 TFA

Size Price Availability Quantity
5mg USD 120  USD120 In stock
10mg USD 200  USD200 In stock
50mg USD 580  USD580 In stock
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Quality Control & Documentation
Biological Activity

β-Casomorphin, human TFA is an opioid-like peptide that is an opioid receptor agonist. Sequence: Tyr-Pro-Phe-Val-Glu-Pro-Ile.

Chemical Information
Molecular Weight 978.02
Formula C46H62F3N7O13
CAS Number 102029-74-3 (free base)
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage -20°C, dry, sealed
Conversion of different model animals based on BSA (PMID: 27057123)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of Compound A used for a mouse (20 mg/kg) to a dose based on the BSA for a rat, multiply 20 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for Compound A of 10 mg/kg.

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Keywords: β-Casomorphin, human TFA, Human β-casomorphin 7 TFA supplier, Opioid Receptor, inhibitors, activators

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