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Bepridil

Cat. No. M30426

All AbMole products are for research use only, cannot be used for human consumption.

Bepridil Structure
Synonym:

(±)-Bepridil; Org 5730

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Quality Control & Documentation
Biological Activity

Bepridil ((±)-Bepridil) is a calcium channel blocking agent used as antiarrhythmic agent. Bepridil inhibits both calcium and sodium currents, has research potential in certain ischemia-induced ventricular arrhythmias. Bepridil also has strong inhibition of SARS-CoV-2 from entry and replication inside Vero E6 and A549 cells.

Chemical Information
Molecular Weight 366.54
Formula C24H34N2O
CAS Number 64706-54-3
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Erol C Vatansever, et al. Proc Natl Acad Sci U S A. Bepridil is potent against SARS-CoV-2 in vitro

[2] F P Zeller, et al. Drug Intell Clin Pharm. Bepridil: a new long-acting calcium channel blocking agent

[3] No authors listed. Lancet. Bepridil

[4] A Gill, et al. Am J Cardiol. Pharmacology of bepridil

[5] L M Hollingshead, et al. Drugs. Bepridil. A review of its pharmacological properties and therapeutic use in stable angina pectoris

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  Catalog
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Keywords: Bepridil, (±)-Bepridil; Org 5730 supplier, Calcium Channel, inhibitors, activators

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