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Anagliptin

Cat. No. M5417

All AbMole products are for research use only, cannot be used for human consumption.

Anagliptin Structure
Synonym:

SK-0403

Size Price Availability
5mg USD 115  USD115 Out of stock
10mg USD 190  USD190 Out of stock
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Quality Control & Documentation
Biological Activity

Anagliptin is a potent and selective DPP-4 inhibitor(IC50= 3.8 nM); > 10 fold less potent for DPP-8 and DPP-9.

Chemical Information
Molecular Weight 383.45
Formula C19H25N7O2
CAS Number 739366-20-2
Solubility (25°C) 36 mg/mL in DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Yang HK, et al. Endocr J. A randomized, placebo-controlled, double-blind, phase 3 trial to evaluate the efficacy and safety of anagliptin in drug-naïve patients with type 2 diabetes.

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Keywords: Anagliptin, SK-0403 supplier, Dipeptidyl Peptidase, inhibitors, activators

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