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Amtolmetin guacil

Cat. No. M30780

All AbMole products are for research use only, cannot be used for human consumption.

Amtolmetin guacil Structure

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Quality Control & Documentation
Biological Activity

Amtolmetin guacil is an effective nonsteroidal anti-Inflammatory agent with pain-relieving effects. Amtolmetin guacil inhibits prostaglandin synthesis and cyclooxygenase (COX). Amtolmetin guacil can stimulate capsaicin receptors present on the gastrointestinal wall and also releases gastroprotective nitric oxide (NO). Amtolmetin guacil can be used to research knee osteoarthritis.

Chemical Information
Molecular Weight 420.46
Formula C24H24N2O5
CAS Number 87344-06-7
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Kunling Wang, et al. Ann Transl Med. Comparison of cardiorenal safety of nonsteroidal anti-inflammatory drugs in the treatment of arthritis: a network meta-analysis

[2] I G Pakhomova. Zh Nevrol Psikhiatr Im S S Korsakova. [A choice of a nonsteroidal anti-inflammatory drug with regard to gastrointestinal and cardiovascular' risks]

[3] Ben-Yong Lou, et al. Acta Crystallogr Sect E Struct Rep Online. 2-Methoxy-phenyl 2-{2-[1-methyl-5-(4-methyl-benzo-yl)pyrrol-2-yl]acetamido}acetate

[4] Kishore Kumar Hotha, et al. Arzneimittelforschung. Species difference in the in vitro and in vivo metabolism of amtolmetin guacil

[5] Kishore Kumar Hotha, et al. Biomed Chromatogr. Validation and clinical application of an LC-ESI-MS/MS method for simultaneous determination of tolmetin and MED5, the metabolites of amtolmetin guacil in human plasma

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Keywords: Amtolmetin guacil supplier, Prostaglandin Receptor, inhibitors, activators

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