Free shipping on all orders over $ 500

Almorexant hydrochloride

Cat. No. M14034

All AbMole products are for research use only, cannot be used for human consumption.

Almorexant hydrochloride Structure
Synonym:

ACT-078573 hydrochloride

Size Price Availability Quantity
1mg USD 55  USD55 In stock
5mg USD 110  USD110 In stock
10mg USD 175  USD175 In stock
25mg USD 350  USD350 In stock
50mg USD 550  USD550 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Almorexant hydrochloride (ACT 078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM, respectively.

Chemical Information
Molecular Weight 549.02
CAS Number 913358-93-7
Solubility (25°C) DMSO ≥ 46 mg/mL
Storage 2-8°C, dry, sealed
References

[1] Michel A Steiner, et al. Neuropsychopharmacology. Differential effects of the dual orexin receptor antagonist almorexant and the GABA(A)-α1 receptor modulator zolpidem, alone or combined with ethanol, on motor performance in the rat

Related OX Receptor Products
CVN766 

CVN766 is an orally active inhibitor of orexin 1 receptor antagonist with blood-brain permeability with the IC50 values of 8 nM and >10 μM for OX1R and OX2R, respectively.

Nivasorexant

Nivasorexant is a potent orexin receptor antagonist.

[Ala11, D-Leu15]-Orexin B(human)

[Ala11,D-Leu15]-Orexin B(human) is a potent and selective orexin-2 receptor (OX2) agonist.

Orexin B, rat, mouse

Orexin B, rat, mouse (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.

Hypocretin (70-98), human

Hypocretin (70-98), human is a polypeptide that is capable of binding to an orexin receptor OX1R and promotes apoptosis.

  Catalog
Abmole Inhibitor Catalog




Keywords: Almorexant hydrochloride, ACT-078573 hydrochloride supplier, OX Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.