Inhibitor/Activator
| Cat.No. | Name | Information |
|---|---|---|
| M5909 | Protirelin | Protirelin is a tripeptide that stimulates the release of thyrotropin and prolactin. Protirelin is a highly conserved neuropeptide that exerts the hormonal control of thyroid-stimulating hormone (TSH) levels as well as neuromodulatory functions. |
| M43608 | Thyroid hormone receptor beta agonist-1 | Thyroid hormone receptor beta agonist-1 is a thyroid beta-agonist. |
| M43607 | THR-β modulator-1 | THR-β modulator-1 is a potent thyroid hormone receptor β modulator. |
| M43606 | THR-β agonist 6 | THR-β agonist 6 is an orally active, selective thyroid hormone receptor β (THR-β) agonist with EC50s of 0.03 μM and 0.22 μM for THR-β and THR-α, respectively. |
| M40979 | TERN-501 | TERN-501 is a thyroid hormone receptor beta (THR-β) agonist that may be used in studies related to non-alcoholic steatohepatitis (NASH). |
| M40748 | ASC41 | ASC41 is a THR-β agonist that can be used in studies related to non-alcoholic steatohepatitis (NASH). |
| M40538 | MBX-2109 | MBX-2109 is a long-acting parathyroid hormone receptor (PTH1R) agonist for studies related to hypoparathyroidism. |
| M29567 | DS08210767 | DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM. |
| M28509 | KB130015 | KB130015 (KB015) is an orally active and potent ThRα and ThRβ (Thyroid Hormone Receptor) inhibitor, with IC50 values of 4.5 and 5.1 μM, respectively. KB130015 has antiarrhythmic properties. KB130015 markedly slows the kinetics of inactivation of Na+ channels. KB130015 opens large-conductance Ca2+-activated K+ channels and relaxes vascular smooth muscle. |
| M27948 | Protirelin acetate | Protirelin Acetate is a highly conserved neuropeptide that exerts the hormonal control of thyroid-stimulating hormone (TSH) levels as well as neuromodulatory functions. |
| M27675 | Taltirelin | Taltirelin (TA0910) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release). |
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