| Cat.No. | Name | Information |
|---|---|---|
| M53460 | SKF107457 | SKF107457 is an HIV-1 protease inhibitor that can be used in AIDS research. |
| M53459 | Mvt-101 | Mvt-101 is a hexapeptide-based inhibitor of HIV-1 protease. |
| M44857 | Ganoderic acid GS-1 | Ganoderic acid GS-1, a highly oxygenated lanostane-type triterpenoid, has anti-HIV-1 protease activities with an IC50 of 58 μM. |
| M41197 | 8-Prenylluteone | 8-Prenylluteone is a HIV-1 protease inhibitor, with an IC50 of 4 μM. |
| M41196 | HIV-1 protease-IN-9 | HIV-1 protease-IN-9 is a HIV-1 protease inhibitor, with a Ki of 0.028 nM. |
| M41195 | HIV-1 protease-IN-12 | HIV-1 protease-IN-12 is a HIV-1 protease inhibitor with an IC50 of 0.51 nM. |
| M41194 | HIV-1 protease-IN-11 | HIV-1 protease-IN-11 is a HIV-1 protease inhibitor with an IC50 of 0.41 nM. |
| M41193 | NNRTIs-IN-3 | NNRTIs-IN-3 is an HIV-1 non-nucleoside reverse transcriptase inhibitor (EC50=0.01 µM). |
| M41192 | HIV-1 protease-IN-8 | HIV-1 protease-IN-8 is a potent HIV-1 protease inhibitor with an IC50 value of 0.32 nM. |
| M40754 | Lenacapavir sodium | Lenacapavir sodium is a first-in-class, long-acting HIV capsid inhibitor. Lenacapavir sodium has anti-HIV activity with an EC50 of 100 pM in MT-4 cells and an average EC50 of 50 pM (20-160 pM) in peripheral blood mononuclear cells against 23 clinical isolates of HIV-1 from different subtypes. |
| M30974 | LEDGIN6 | LEDGIN6 (CX05168) is a quinoline-based protein-protein interaction inhibitor of LEDGF/p75 and HIV integrase. |
| M30871 | Tenofovir exalidex | Tenofovir exalidex (CMX157) is a lipid conjugate of the acyclic nucleotide analog Tenofovir with activity against both wild-type and antiretroviral drug-resistant HIV strains, including multidrug nucleoside/nucleotide analog-resistant viruses. Tenofovir exalidex is active against all major subtypes of HIV-1 and HIV-2 in fresh human PBMCs and against all HIV-1 strains evaluated in monocyte-derived macrophages, with EC50s ranging between 0.2 and 7.2 nM. CMX157 is orally available and has no apparent toxicity. Tenofovir exalidex also shows antiviral activity against HBV. |
| M30742 | Islatravir | Islatravir (MK-8591) is a potent anti-HIV-1 agent, acting as a nucleoside reverse transcriptase inhibitor, with EC50s of 0.068 nM, 3.1 nM and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively. |
| M30740 | Fostemsavir Tris | Fostemsavir Tris (BMS-663068 (Tris)) is the phosphonooxymethyl proagent of BMS-626529. Fostemsavir Tris (BMS-663068 (Tris)) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells. |
| M30708 | Patentiflorin A | Patentiflorin A is a potent, broadspectrum HIV-1 inhibitor. Patentiflorin A also inhibits HIV drug-resistant strains. |
| M30693 | SAMT-247 | SAMT-247 is a microbicide that selectively inactivate the viral nucleocapsid protein NCp7, causing zinc ejection and preventing RNA encapsidation. SAMT-247 shows good antiviral activity. |
| M30530 | Ilimaquinone | Ilimaquinone, a marine sponge metabolite, displays anticancer activity via GADD153-mediated pathway. Ilimaquinone can induce vesiculation of the Golgi apparatus. Ilimaquinone exerts anti-HIV, anti-microbial, anti-inflammatory, and effects. |
| M30463 | Formycin A | Formycin A (NSC 102811), a purine nucleoside antibiotic, is a potent human immunodeficiency virus type 1 (HIV-1) inhibitor with an EC50 of 10 μM. Formycin A shows antitumor and antiviral activities. |
| M30402 | Censavudine | Censavudine (OBP-601; BMS-986001), a nucleoside analog, is a nucleoside reverse transcriptase inhibitor. Censavudine is a potent HIV inhibitor with EC50 ranges from 30 nM to 81 nM and 450 nM to 890 nM for HIV-2 and HIV-1, respectively. |
| M30378 | BMS-585248 | BMS-585248 is a potent, third-generation HIV-1 attachment inhibitor with a promising initial in vitro and in vivo pharmacokinetic profile. |
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