About 1 result found for searched term "Relacatib" (0.125 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M29991 | Relacatib | Cathepsin |
| SB-462795 | ||
| Relacatib (SB-462795) is a novel, potent, and orally active inhibitor of human cathepsins K, L, and V with Ki values of 41 pM, 68 pM, and 53 pM, respectively. Relacatib inhibits endogenous cathepsin K in situ in human osteoclasts and human osteoclast-mediated bone resorption with IC50 values of 45 nM and 70 nM, respectively. Relacatib inhibits bone resorption in vitro in human tissue as well as in cynomolgus monkeys in vivo. | ||
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