About 7 results found for searched term "Orexin receptor antagonist 3" (0.129 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M14037 | Orexin receptor antagonist 3 | OX Receptor |
| Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist. | ||
| M3261 | Almorexant | OX Receptor |
| ACT-078573 | ||
| Almorexant is a competitive OX1 and OX2 orexin receptor antagonist with IC50 of 13 and 8 nM, respectively. | ||
| M3760 | TCS-1102 | OX Receptor |
| TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively). | ||
| M10955 | Nemorexant | OX Receptor |
| ACT-541468 | ||
| Nemorexant (ACT-541468) is an effective orexin receptor antagonist. It also has IC50s of 2 nM and 3 nM for the Ox1 receptor and Ox2 receptor, respectively. | ||
| M14034 | Almorexant hydrochloride | OX Receptor |
| ACT-078573 hydrochloride | ||
| Almorexant hydrochloride (ACT 078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM, respectively. | ||
| M14035 | EMPA | OX Receptor |
| EMPA is a high-affinity, reversible and selective orexin OX2 receptor antagonist. [3H]EMPA binds to human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM respectively. | ||
| M40751 | Nemorexant hydrochloride | OX Receptor |
| Nemorexant hydrochloride is an orally active dual orexin type 1 and type 2 (OX1 and OX2) receptor antagonist (DORA) as well as an inhibitor of BCRP, with an IC50 value of 3.0 μM when acting on BCRP, and can be used in studies related to insomnia. | ||
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