About 30 results found for searched term "Opioid Receptor" (0.072 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M1953 | ADL5859 Hydrochloride | Opioid Receptor |
| ADL5859 HCl | ||
| ADL5859 is a potent, selective and orally bioavailable δ-opioid receptor agonist (Ki = 0.84 nM, EC50 = 20 nM). | ||
| M2145 | Loperamide hydrochloride | Animal Modeling |
| R-18553 hydrochloride | ||
| Loperamide hydrochloride is a high affinity μ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for μ-, δ- and κ-opioid receptors respectively. Loperamide hydrochloride is also a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. It can be used to construct animal models of functional constipation. | ||
| M2214 | JTC-801 | Opioid Receptor |
| JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM. | ||
| M2875 | Nalmefene hydrochloride | Opioid Receptor |
| Nalmefene is an opioid receptor antagonist, it is used primarily in the management of alcohol dependence. | ||
| M2991 | Cutamesine dihydrochloride | Sigma Receptor |
| AGY94806 dihydrochloride; SA 4503 dihydrochloride | ||
| Cutamesine dihydrochloride (SA4503 dihydrochloride; AGY94806 dihydrochloride) is a novel and selective opioid sigma1 receptor agonist with IC50 of 17.4 nM. | ||
| M1577 | Naltrexone Hydrochloride | Opioid Receptor |
| Naltrexone hydrochlorideis an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence. | ||
| M4456 | Sec-O-Glucosylhamaudol | Opioid Receptor |
| Sec-o-glucosylhamaudol is a natural product isolated from The apostrophophore, which can reduce the protein level of μ-opioid receptor and can be used for pain relief research. | ||
| M4516 | Sinomenine-Hydrochloride | NF-κB |
| Cucoline hydrochloride | ||
| Sinomenine hydrochloride (Cucoline hydrochloride), an alkaloid derived from Sinomenium Acutum, is a blocker of NF-κB activation. Sinomenine is also a μ-opioid receptor activator. | ||
| M4520 | (+)-Corydaline | AChR/AChE |
| (+)-Corydaline; Corydalin | ||
| Corydaline ((+) -corydaline) is an isoquinoline alkaloid extracted from Corydalis Yanhusuo. It is an inhibitor of AChE with IC50 of 226 µM. Corydaline is a μ-opioid receptor agonist (Ki = 1.23 µM) that inhibits the replication of enterovirus 71 (EV71) (IC50 = 25.23 µM). Corydaline has anti-angiogenesis, anti-allergy, gastric emptying and anti-nociception effects. | ||
| M4808 | TRV130 hydrochloride | Opioid Receptor |
| Oliceridine HCl; TRV130 HCl | ||
| TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand. | ||
| M5065 | Cebranopadol | Opioid Receptor |
| GRT-6005 | ||
| Cebranopadol is a NOP and opioid receptor agonist that acts on human NOP, MOP, KOP and δ-opioid peptide (DOP) receptors with Ki/EC50 values of 0.9 nM/13 nM and 0.7 nM/1.2 nM, respectively. 2.6 nM/17 nM, 18 nM/110 nM. | ||
| M5067 | Eluxadoline | Others |
| Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist. | ||
| M5289 | PZM21 | Opioid Receptor |
| PZM21 is a potent and selective μ-opioid-receptor (μOR) agonist with an EC50 of 1.8 nM. | ||
| M5403 | Alvimopan dihydrate | Opioid Receptor |
| LY 246736 dihydrate; ADL 8-2698 dihydrate | ||
| Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). | ||
| M7314 | SNC 80 | Opioid Receptor |
| NIH 10815; SNC80 | ||
| SNC 80 is a highly selective non-peptide δ-opioid receptor agonist with a Ki of 1.78 nM and an IC50 of 2.73 nM. | ||
| M7882 | Levallorphan tartrate salt | Others |
| Partial agonist (antagonist) at μ and δ opioid receptors. | ||
| M7946 | Naloxone methiodide | Others |
| Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors. | ||
| M7951 | Naltrindole isothiocyanate hydrochloride | Others |
| Naltrindole isothiocyanate hydrochloride is a selective irreversible δ2 opioid receptor antagonist. | ||
| M7984 | Opipramol dihydrochloride | Others |
| σ1/σ2 opioid receptor agonist; an antagonist at D2, 5HT2 and H1 receptors; atypical antidepressant, antipsychotic and anxiolytic. | ||
| M8030 | PB28 dihydrochloride | Others |
| Selective σ2 opioid receptor ligand; putative σ2 agonist. | ||
| M8191 | Salvinorin A | Others |
| Salvinorin A is a potent, non-nitrogenous κ opioid selective receptor agonist. | ||
| M8453 | ML138 | Others |
| ML138 (CID 44601470) is a highly selective agonist at kappa opioid receptors (KOR) that potently activate G protein coupling but weakly interact with β arrestin2. | ||
| M8502 | Alvimopan | Opioid Receptor |
| ADL 8-2698; LY 246736 | ||
| Alvimopan is a gastroprokinetic peripheral mu-opioid receptor antagonist. | ||
| M8776 | ARM390 | Others |
| ARM390 in a δ-selective opioid receptor agonist derivative of SNC80. | ||
| M8832 | U-69593 | Opioid Receptor |
| U69593 | ||
| U-69593 is a selective κ opioid receptor agonist. | ||
| M8834 | U-62066 | Others |
| Highly selective κ opioid receptor agonist; antitussive. | ||
| M9268 | Met-Enkephalin | Opioid Receptor |
| H-Tyr-Gly-Gly-Phe-Met-OH; Methionine enkephalin; Metenkefalin | ||
| Met-Enkephalin (H-Tyr-Gly-Gly-Phe-Met-OH) inhibits tumor growth via binding to the opioid receptor. | ||
| M9514 | JDTic | Opioid Receptor |
| JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects. | ||
| M9615 | DAMGO | Opioid Receptor |
| RX783006; Dagol | ||
| DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. | ||
| M10229 | Porcine dynorphin A (1-13) | Opioid Receptor |
| Dynorphin A Porcine Fragment 1-13 | ||
| Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist. | ||
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