About 5 results found for searched term "NMDA receptor antagonist 7" (0.129 seconds)
Cat.No. | Name | Target |
---|---|---|
M42201 | NMDA receptor antagonist 7 | GluR |
NMDA receptor antagonist 7 is GluN2B subunit-selective NMDA Receptor antagonist, with an Ki of 93 nM and an IC50 of 72 nM. | ||
M7581 | Dizocilpine maleate | NMDA |
Dizocilpine hydrogen maleate; (+)-MK 801 maleate; MK-801 maleate | ||
Dizocilpine maleate (MK-801 maleate) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes. | ||
M30021 | DQP-1105 | GluR |
DQP-1105 is a potent noncompetitive NMDA receptor antagonist. DQP-1105 inhibits GluN2C- and GluN2D-containing receptors (IC50=7.0 and 2.7 μM, respectively). The IC50 values are at least 50-fold lower than those for recombinant GluN2A-, GluN2B-, GluA1-, or GluK2-containing receptors. | ||
M56508 | SDZ 220-581 | GluR |
SDZ 220-581 is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. | ||
M56498 | SDZ 220-581 Ammonium salt | GluR |
SDZ 220-581 Ammonium salt is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. |
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