About 30 results found for searched term "Histamine Receptor" (0.059 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2398 | Antazoline hydrochloride | Histamine Receptor |
| Phenazoline hydrochloride | ||
| Antazoline hydrochloride is a first generation antihistamine, binding to the histamine H1 receptor and blocking the action of endogenous histamine. | ||
| M2449 | Bepotastine Besilate | Histamine Receptor |
| Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7. | ||
| M2452 | Betahistine dihydrochloride | Histamine Receptor |
| Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM. | ||
| M2545 | Cyclizine dihydrochloride | Histamine Receptor |
| Cyclizine 2HCl is a piperazine derivative with Histamine H1 receptor antagonist activity. | ||
| M2582 | Clemizole | Histamine Receptor |
| Clemizole is a H1 histamine receptor antagonist with IC50 Value of 8 mM (NS4B). | ||
| M2621 | Desloratadine | Histamine Receptor |
| Sch34117 | ||
| Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM. | ||
| M2639 | Dimaprit dihydrochloride | Histamine Receptor |
| Dimaprit is a histamine type 2 receptor agonist. | ||
| M2643 | Diphenylpyraline hydrochloride | Histamine Receptor |
| 4-Diphenylmethoxy-1-methylpiperidine hydrochloride | ||
| Diphenylpyraline hydrochloride (DPP) is an internationally available antihistamine that produces therapeutic antiallergic effects by binding to histamine H₁ receptors. | ||
| M2650 | Doxepin hydrochloride | Histamine Receptor |
| Doxepin hydrochloride is a potent and selective histamine receptor H1 antagonist. Doxepin hydrochloride is also a potent CYP450 inhibitor and significantly inhibits CYP450 2C19 and 1A2. | ||
| M2653 | Doxylamine Succinate | Histamine Receptor |
| Doxylamine succinate competitively inhibits histamine at H1 receptors with substantial sedative and anticholinergic effects. | ||
| M2660 | Ebastine | Histamine Receptor |
| LAS-W 090; RP64305 | ||
| Ebastinea is an orally active, potent histamine H1 receptor antagonist for studies related to allergic diseases. | ||
| M2671 | Epinastine hydrochloride | Histamine Receptor |
| WAL801 hydrochloride | ||
| Epinastine hydrochloride is an antihistamine and mast cell stabilizer. Epinastine hydrochloride is a potent, selective and orally-active histamine H1 receptor antagonist. | ||
| M2699 | Fexofenadine hydrochloride | Histamine Receptor |
| MDL 16455A | ||
| Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM. | ||
| M2755 | Histamine Phosphate | Histamine Receptor |
| Histamine diphosphate | ||
| Histamine Phosphate is an endogenous ligand for the histamine receptor that can induce allergic reactions by acting with H1 receptors, promote acid secretion by acting with H2 receptors, and inhibit histamine release and modulate immune responses by acting with H3 receptors and H4 receptors. It can be used in studies related to allergy, hyperacidity, sleep disorders, asthma and many other diseases. | ||
| M2756 | Histamine dihydrochloride | Histamine Receptor |
| Histamine 2HCl is an endogenous ligand for the histamine receptor, which can cause allergic reactions by interacting with H1 receptors, promote acid secretion by interacting with H2 receptors, as well as inhibit histamine release and modulate immune responses by interacting with H3 receptors and H4 receptors. It can be used in studies related to allergy, hyperacidity, sleep disorders, asthma and many other diseases. | ||
| M2760 | Hydroxyzine dihydrochloride | Histamine Receptor |
| Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM. | ||
| M2784 | JNJ-7777120 | Histamine Receptor |
| JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM, exhibits >1000-fold selectivity over the other histamin receptors. | ||
| M2811 | Levodropropizine | Histamine Receptor |
| (S)-(-)-Dropropizine | ||
| Levodropropizine possess anti-allergic and inhibits histamine receptor, reduces cough by interfering with stimulus activation of peripheral endings of sensory nerves and by modulation of neuropeptides involved in the cough reflex. | ||
| M2971 | Pyrilamine Maleate | Histamine Receptor |
| Mepyramine Maleate | ||
| Pyrilamine is a histamine H1 receptor inverse agonist, it binds to a G protein-coupled form of the receptor and promotes a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11-mediated signaling. | ||
| M2990 | Rupatadine Fumarate | Histamine Receptor |
| Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively. | ||
| M3213 | Meclizine dihydrochloride | Histamine Receptor |
| Meclozine dihydrochloride; NSC28728 | ||
| Meclizine is a histamine H1 receptor antagonist used to treat nausea and motion sickness, has anti-histamine, anti-muscarinic and anti-oxidative phosphorylation properties, also an agonist ligand for mCAR (constitutive androstane receptor) and an inverse agonist for hCAR. Phase2. | ||
| M3226 | Brompheniramine hydrogen maleate | Histamine Receptor |
| Brompheniramine hydrogen maleate is a histamine H1 receptors antagonist. | ||
| M3318 | Clemastine Fumarate | Histamine Receptor |
| Meclastine fumarate | ||
| Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM. | ||
| M3383 | Diphenhydramine hydrochloride | Histamine Receptor |
| DPH | ||
| Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB). | ||
| M3385 | Cimetidine | Histamine Receptor |
| SKF-92334 | ||
| Cimetidine, a histamine congener, competitively inhibits histamine binding to histamine H2 receptors. | ||
| M3431 | Nizatidine | Histamine Receptor |
| Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM. | ||
| M3458 | Chlorpheniramine Maleate | Histamine Receptor |
| Chlorphenamine maleate | ||
| Chlorpheniramine (Chlorpheniramine maleate, Chlorphenamine) is an histamine H1 receptor antagonist with IC50 of 12 nM. | ||
| M3592 | Chlorprothixene | Dopamine Receptor |
| Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively. | ||
| M3665 | Promethazine hydrochloride | Histamine Receptor |
| Promethazine hydrochloride is a potent histamine H1 receptor antagonist used as a sedative and antiallergic compound. | ||
| M5393 | Alcaftadine | Histamine Receptor |
| Lastacaft, R89674, R 89674, R-89674 | ||
| Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines. Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor. | ||
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