About 17 results found for searched term "Eph-inhibitor-1" (0.141 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M20738 | Eph-inhibitor-1 | Ephrin Receptor |
| Eph inhibitor 2 | ||
| Eph-inhibitor-1 (Eph inhibitor 2) is an Eph family tyrosine kinase inhibitor that targets Eph receptors. | ||
| M43494 | Eph inhibitor 1 | Ephrin Receptor |
| Eph inhibitor 1 is a potent Eph inhibitor. | ||
| M2408 | Atomoxetine hydrochloride | 5-HT Receptor |
| Tomoxetine hydrochloride; LY 139603; (R)-Tomoxetine hydrochloride | ||
| Atomoxetine is a selective norepinephrine (NE) transporter inhibitor with Ki of 5 nM, with 15- and 290-fold lower affinity for human 5-HT and DA transporters. | ||
| M3582 | Racecadotril | Neprilysin (NEP) |
| Acetorphan | ||
| Racecadotril is a peripheral enkephalinase inhibitor with an IC50 of 4.5 μM.Racecadotril and its active metabolite, Thiorphan, inhibited the activity of purified NEP in the mouse brain with Ki's of 4500 and 6.1 nM.May be used in diarrhea related studies. | ||
| M7949 | Nisoxetine hydrochloride | Others |
| Nisoxetine hydrochloride is a potent, selective norepinephrine transporter inhibitor (Ki = 5.1 nM). | ||
| M8509 | Sephin1 | Others |
| Sephin1 (selective inhibitor of a holophosphatase) is a guanabez derivative that binds to and inhibits a regulatory subunit of the stress-induced protein phosphatase 1 (PPP1R15A), but not the constitutive PPP1R15B, and lacks ?2-adrenergic activity. | ||
| M8974 | ALW-II-41-27 | Ephrin Receptor |
| Eph receptor tyrosine kinase inhibitor | ||
| ALW-II-41-27 is a Eph receptor tyrosine kinase inhibitor with an IC50 of 11 nM for EPHA2. | ||
| M9823 | Cephalosporin C zinc salt | Others |
| Cephalosporin C zinc salt is a potent SAMHD1 inhibitor, with IC50 of 1.1 μM. | ||
| M27759 | Cefepime hydrochloride | Antibiotic |
| BMY-28142 hydrochloride | ||
| Cefepime hydrochloride is a cephalosporin antibiotic agent. Cefepime hydrochloride has inhibitory activity against human serum paraoxonase-1 (hPON1) with an IC50 value of 21.115 mM. | ||
| M28151 | (E/Z)-Icerguastat | Phosphatase |
| (E/Z)-Sephin1; (E/Z)-IFB-088 | ||
| (E/Z)-Icerguastat ((E/Z)-Sephin1) is a selective inhibitor of the phosphatase regulatory subunit PPP1R15A (R15A). (E/Z)-Icerguastat can be used for protein misfolding diseases research. | ||
| M30309 | Setiptiline | 5-HT Receptor |
| Org-8282 | ||
| Setiptiline (Org-8282) is a serotonin receptor antagonist. Setiptiline is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine. | ||
| M30707 | Setiptiline maleate | 5-HT Receptor |
| MO-8282 | ||
| Setiptiline maleate (MO-8282 maleate) is a serotonin receptor antagonist. Setiptiline maleate is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline maleate acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine. | ||
| M40568 | Apicularen B | ATPase |
| Apicularen B is a cytotoxic macrolide produced by Archangium gephyra and is also a specific V-ATPase inhibitor. Its IC50 values range from 0.2 to 1.2 μg/mL and it exhibits weak activity against some Gram-positive bacteria. | ||
| M49949 | LDN-211904 oxalate | Ephrin Receptor |
| LDN-211904 oxalate is a potent and selective EphB3 inhibitor with an IC50 of 0.079 µM.LDN-211904 oxalate showed good metabolic stability in mouse liver microsomes.LDN-211904 oxalate was shown to be effective in inhibiting STAT3-activated CSC stemness in combination with cetuximab. | ||
| M56733 | Icerguastat Carbonate | Phosphatase |
| Icerguastat (Sephin1) Carbonate, a derivative of Guanabenz lacking the α2-adrenergic activity, is a selective inhibitor of the phosphatase regulatory subunit PPP1R15A (R15A). | ||
| M56091 | Tedatioxetine | 5-HT Receptor |
| Tedatioxetine (Lu AA24530) acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist. | ||
| M56076 | Tedatioxetine hydrobromide | 5-HT Receptor |
| Tedatioxetine (Lu AA24530) hydrobromide acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist. | ||
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