ERK1/2 inhibitor 1 - Search Results

About 9 results found for searched term "ERK1/2 inhibitor 1" (0.128 seconds)

Cat.No.	Name	Target
M14152	ERK1/2 inhibitor 1	ERK
	ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.
M10741	ERK1/2 inhibitor 2	ERK
	ERK1/2 inhibitor 2 (Example 1) is a potent dual ERK1/2 inhibitor. ERK1/2 inhibitor 2 has anti-cancer activity.
M11529	Temuterkib	ERK
	LY3214996
	Temuterkib (LY3214996) is a selective, novel erK1/2 inhibitor with an IC50 of 5 nM against ERK1 and ERK2. It can effectively inhibit intracellular P-RSK1 in cancer cell lines with BRAF and RAS mutations. Temuterkib has strong antitumor activity in cancer models with altered MAPK pathways.
M42119	ERK1/2 inhibitor 9	ERK
	ERK1/2 inhibitor 9 (Probe 1) is a covalent ERK1/2 inhibitor.
M49701	ERK1/2 inhibitor 3	ERK
	ERK1/2 inhibitor 3 is a potent inhibitor of ERK1/2.
M49702	ERK1/2 inhibitor 4	ERK
	ERK1/2 inhibitor 5 is a potent inhibitor of ERK1/2.
M49703	ERK1/2 inhibitor 5	ERK
	ERK1/2 inhibitor 5 is a potent inhibitor of ERK1/2.
M49704	ERK1/2 inhibitor 6	ERK
	ERK1/2 inhibitor 6 is a potent inhibitor of ERK1/2.
M49720	STE-MEK1(13)	ERK
	STE-MEK1(13) (Ste-MPKKKPTPIQLNP-NH?) is a cell permeable ERK1/2 inhibitor (IC50: 13-30?μM).