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 About 6 results found for searched term "Adenosine Receptor" (0.054 seconds)

Cat.No.  Name Target
M8825 Adenosine A1 receptor activator T62 Adenosine Receptor
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor.
M40652 Adenosine receptor antagonist 2 Adenosine Receptor
Adenosine receptor antagonist 2 is a potent, orally active and antitumor active adenosine receptor A2a/A2b antagonist with IC50 values of 1 nM and 3 nM, respectively.
M40660 Adenosine receptor antagonist 1 Adenosine Receptor
Adenosine receptor antagonist 1 is a selective adenosine receptor A2aR antagonist with an IC50 value of 0.29 nM and a 14-fold higher selectivity for A2aR than for A2bR.
M40661 Adenosine receptor inhibitor 2 Adenosine Receptor
Adenosine receptor inhibitor 2 is a potent adenosine receptor AR inhibitor with dual affinity for A1/A2A ARs with Ki values of 52.2 and 167 nM, respectively.
M40664 Adenosine receptor inhibitor 1 Adenosine Receptor
Adenosine receptor inhibitor 1 is a potent, selective adenosine receptor inhibitor with Ki values of >1000, 68.5, >1000, >1000, >1000 nM for A1AR, A2AAR, A2BAR, and A3AR, respectively, and possesses analgesic as well as anti-inflammatory activity. It has analgesic and anti-inflammatory activities and can be used in cancer and neurodegenerative disease research.
M41759 Adenosine receptor antagonist 4 Adenosine Receptor
Adenosine receptor antagonist 4 is an adenosine A1 receptor antagonist with a Ki of 101 nM for human A1 receptor.



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