About 6 results found for searched term "Adenosine Receptor" (0.054 seconds)
Cat.No. | Name | Target |
---|---|---|
M8825 | Adenosine A1 receptor activator T62 | Adenosine Receptor |
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor. | ||
M40652 | Adenosine receptor antagonist 2 | Adenosine Receptor |
Adenosine receptor antagonist 2 is a potent, orally active and antitumor active adenosine receptor A2a/A2b antagonist with IC50 values of 1 nM and 3 nM, respectively. | ||
M40660 | Adenosine receptor antagonist 1 | Adenosine Receptor |
Adenosine receptor antagonist 1 is a selective adenosine receptor A2aR antagonist with an IC50 value of 0.29 nM and a 14-fold higher selectivity for A2aR than for A2bR. | ||
M40661 | Adenosine receptor inhibitor 2 | Adenosine Receptor |
Adenosine receptor inhibitor 2 is a potent adenosine receptor AR inhibitor with dual affinity for A1/A2A ARs with Ki values of 52.2 and 167 nM, respectively. | ||
M40664 | Adenosine receptor inhibitor 1 | Adenosine Receptor |
Adenosine receptor inhibitor 1 is a potent, selective adenosine receptor inhibitor with Ki values of >1000, 68.5, >1000, >1000, >1000 nM for A1AR, A2AAR, A2BAR, and A3AR, respectively, and possesses analgesic as well as anti-inflammatory activity. It has analgesic and anti-inflammatory activities and can be used in cancer and neurodegenerative disease research. | ||
M41759 | Adenosine receptor antagonist 4 | Adenosine Receptor |
Adenosine receptor antagonist 4 is an adenosine A1 receptor antagonist with a Ki of 101 nM for human A1 receptor. |
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