About 4 results found for searched term "Acetylcholine Chloride" (0.125 seconds)
Cat.No. | Name | Target |
---|---|---|
M3317 | Acetylcholine Chloride | AChR/AChE |
Ach; ACh chloride | ||
The chemical compound Acetylcholine Chloride is a neurotransmitter in both the peripheral nervous system (PNS) and central nervous system (CNS) in many organisms including humans. | ||
M9058 | Varenicline hydrochloride | AChR/AChE |
CP 526555 hcl; Chantix; Champix | ||
Varenicline hydrochloride is a potent partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR, with EC50s of 2.3 μM and 55 μM, respectively. In addition, Varenicline hydrochloride is also a potent full agonist of α7 nAChRs. In addition, Varenicline hydrochloride is a potent full α7 nAChRs agonist with an EC50 of 18 μM. | ||
M20984 | Varenicline dihydrochloride | AChR/AChE |
Chantix, Champix | ||
Varenicline (CP 526555, Chantix, Champix) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation. | ||
M30563 | Anagyrine hydrochloride | AChR/AChE |
(-)-Anagyrine hydrochloride; Monolupine hydrochloride; Rhombinine hydrochloride | ||
Anagyrine ((-)-Anagyrine) hydrochloride is a quinolizidine alkaloid that has been found in Lupinus albus. Anagyrine hydrochloride binds to muscarinic and nicotinic acetylcholine receptors with IC50 values of 132 and 2096 µM respectively. Anagyrine hydrochloride is a potent and effective desensitizer of nAChR, and Anagyrine hydrochloride can directly, without metabolism, desensitize nAChR. |
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