About 7 results found for searched term "A2A receptor antagonist 3" (0.13 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M40663 | A2A receptor antagonist 3 | Adenosine Receptor |
| A2A receptor antagonist 3 is an adenosine receptor A2a antagonist with a Ki of 0.4 nM. It binds to A2b, A1, and A3 receptors with Ki values of 37, 107, and 1467 nM, respectively. | ||
| M6920 | Lu AA 47070 | Others |
| Lu AA 47070 is a potent and selective precursor compound of adenosine A2A receptor antagonists with Ki values of 5.9, 260, 410 and <10,000 nM for A2A, A2B, A1 and A3 receptors, respectively. | ||
| M10191 | Vipadenant | Adenosine Receptor |
| BIIB014; CEB-4520 | ||
| Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. | ||
| M30180 | ST 1535 | Adenosine Receptor |
| ST 1535 is a potent and orally active A2A adenosine receptor antagonist. ST 1535 shows antiparkinsonian activity and antitremorigenic effects. ST 1535 has the potential for the research of Parkinson’s disease. | ||
| M40653 | A2AR-antagonist-1 | Adenosine Receptor |
| A2AR-antagonist-1 is an orally active adenosine receptor A2AR antagonist with an IC50 value of 29 nM.A2AR-antagonist-1 is also a T-cell activator that acts by inhibiting immunosuppressive molecules (LAG-3 and TIM-3) and potentiating effector molecules (GZMB, IFNG and IL-2). It has antitumor activity and is metabolically stable in mouse liver microsomes. | ||
| M40659 | hA2A/hCA XII modulator 1 | Adenosine Receptor |
| hA2A/hCA XII modulator 1 is a triazolopyrazine and a potent adenosine receptor hA2A antagonist, with Ki of 6.4 nM, 4.819 μM, and >30 μM for hA2AAR, hA1AR, and hA3AR, respectively. hA2A/hCA XII modulator 1 is a potent inhibitor of human carbonic anhydrase XII (hCA XII). In addition, hA2A/hCA XII modulator 1 is also a potent human carbonic anhydrase XII (hCA XII) inhibitor with Ki of 6.2 nM, 46 nM, 466 nM, 8.351 μM for hCA XII, hCA II, hCA IX, and hCA I, respectively, and can be used in cancer-related studies. | ||
| M40667 | A2A receptor antagonist 2 | Adenosine Receptor |
| A2A receptor antagonist 2 is a potent, highly selective adenosine receptor A2A antagonist with an IC50 value of 8.3 nM. | ||
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