About 9 results found for searched term "53-85-0" (0.183 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M5321 | CX-6258 HCl | Pim |
| CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3, respectively. | ||
| M17520 | Desoxo-narchinol A | Sesquiterpenoids |
| Desoxo-narchinol A | ||
| M31193 | 5,6-Dichlorobenzimidazole riboside | CDK |
| 5,6-Dichlorobenzimidazole riboside is a nucleoside analog that inhibits several carboxyl-terminal domain (CTD) kinases including casein kinase II and CDKs. 5,6-Dichlorobenzimidazole riboside trigger p53-dependent apoptosis of human colon adenocarcinoma cells without inducing genotoxic stress to healthy cells. | ||
| M43703 | Thaumatins | Others |
| Thaumatins is a protein, which can be purified from the fruit of Thaumatococcus daniellii Benth. | ||
| M8930 | EMD534085 | Kinesin |
| EMD534085 is a potent and selective inhibitor of the mitotic kinesin-5 with an IC50 of 8 nM. | ||
| M10253 | Ralinepag | Prostaglandin Receptor |
| APD811 | ||
| Ralinepag (APD811) is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist with EC50 of 8.5 nM, 530 nM and 850 nM for human IP receptor, rat IP receptor and human DP1 receptor, respectively. | ||
| M28966 | CB-5339 | p97 |
| CB-5339 is a potent p97 inhibitor with an IC50 <30 nM (WO2015109285A1, compound FF07). | ||
| M29784 | DS45500853 | Estrogen Receptor |
| DS45500853 is an estrogen-related receptor α (ERRα) agonist. DS45500853 inhibits the binding between receptor-interacting protein 140 (RIP140) corepressor peptide (10 nM) and GST-ERRα ligand-binding domain (LBD; 1.2 μM) with an IC50 value of 0.80 μM. DS45500853 can be used for the research of metabolic disorders, including type 2 diabetes mellitus (T2DM). | ||
| M30755 | ONO-5334 | Cathepsin |
| ONO-5334 is a potent, selective and orally active cathepsin K inhibitor with Ki values of 0.10 nM, 0.049 nM and 0.85 nM for human, rabbit and rat cathepsin K, respectively. ONO 5334 is an effective antiviral compound against SAR-COV-2 virus activity with an EC50 value of 500 nM. ONO-5334 has the potential for the study of osteoporosis and COVID-19 disease. | ||
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