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Seralutinib (GB002)

Cat. No. M20835

All AbMole products are for research use only, cannot be used for human consumption.

Seralutinib (GB002) Structure
Synonym:

PK10571

Size Price Availability Quantity
5mg USD 120  USD120 In stock
10mg USD 180  USD180 In stock
25mg USD 320  USD320 In stock
50mg USD 420  USD420 In stock
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Quality Control & Documentation
Biological Activity

Seralutinib (PK10571, GB002) is a novel PDGFR kinase inhibitor with IC50s of 8 nM and 10 nM for PDGFRα and PDGFRβ in enzyme assays, respectively.

Chemical Information
Molecular Weight 469.54
Formula C27H27N5O3
CAS Number 1619931-27-9
Solubility (25°C) DMSO 94 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Robert P Frantz, et al. Pulm Circ. TORREY, a Phase 2 study to evaluate the efficacy and safety of inhaled seralutinib for the treatment of pulmonary arterial hypertension

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  Catalog
Abmole Inhibitor Catalog




Keywords: Seralutinib (GB002), PK10571 supplier, VEGFR/PDGFR, inhibitors, activators

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