(S,S)-GSK321

Cat. No. M54536

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(S,S)-GSK321 is the (S,S)-enantiomer of GSK321.GSK321 is a potent inhibitor of the mutant isocitrate dehydrogenase 1 (IDH1) enzyme.

Related Isocitrate Dehydrogenase (IDH) Products
Mutant IDH1-IN-4 Mutant IDH1-IN-4 is an inhibitor of mutant isocitrate dehydrogenase 1 (IDH 1) with an IC50 value of ≤ 0.5 μM for mutant IDH 1 in R132H, HT1080 and U87R132H cells.
IDH1 Inhibitor 1 IDH1 Inhibitor 1 is a potent, orally bioavailable, brain-permeable, selective mutant IDH1 inhibitor that inhibits IDH1R132H, IDH1R132C, and IDH1WT with IC50s of 0.021 μM, 0.045 μM, and 2.52 μM, respectively. possesses antitumor activity.
IDH1 Inhibitor 7 IDH1 Inhibitor 7 is an IDH1 inhibitor with an IC50 of less than 100 nM.
(R,R)-GSK321 (R,R)-GSK321 is an isomer of GSK321 and a wild-type isocitrate dehydrogenase 1 (WT IDH1) inhibitor with an IC50 value of 120 nM.
IDH1 Inhibitor 2 IDH1 Inhibitor 2 is a potent wild-type IDH1 inhibitor that acts through covalent modification of His315 and has an IC50 value of 110 nM.

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