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Pegdinetanib

Cat. No. M25278

All AbMole products are for research use only, cannot be used for human consumption.

Pegdinetanib Structure
Synonym:

BMS-844203; CT-322

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Quality Control & Documentation
Biological Activity

Pegdinetanib (BMS-844203; CT-322) is a selective VEGFR-2 (VEGFR) inhibitor with Kds of 11 nM and 250 nM and IC50s of 16 nM and 240 nM for human and murine VEGFR-2, respectively. Pegdinetanib does not bind to VEGFR-1 or VEGFR-3. Pegdinetanib has antitumor activity.

Chemical Information
CAS Number 906450-24-6
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
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  Catalog
Abmole Inhibitor Catalog




Keywords: Pegdinetanib, BMS-844203; CT-322 supplier, VEGFR/PDGFR, inhibitors, activators

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