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PD 173212

Cat. No. M7106

All AbMole products are for research use only, cannot be used for human consumption.

PD 173212 Structure
Synonym:

PD173212

Size Price Availability Quantity
2mg USD 80  USD80 In stock
5mg USD 150  USD150 In stock
10mg USD 240  USD240 In stock
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Quality Control & Documentation
Biological Activity

PD 173212 is a potent N-type voltage-gated calcium channel blocker (IC50 = 36 nM). PD 173212 displays selectivity over K+, Na+ and L-type Ca2+ channels. PD 173212 prevents tonic seizures in the audiogenic seizure model in vivo.

Chemical Information
Molecular Weight 599.85
Formula C38H53N3O3
CAS Number 217171-01-2
Solubility (25°C) DMSO 59.98 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Deng, et al. Neuropharmacology. Huwentoxin-XVI, an analgesic, highly reversible mammalian N-type calcium channel antagonist from Chinese tarantula Ornithoctonus huwena.

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Keywords: PD 173212, PD173212 supplier, Calcium Channel, inhibitors, activators

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