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NNC 55-0396 dihydrochloride is a highly selective T-type calcium channel blocker. Displays IC50 values of 6.8 and > 100 μM for inhibition of Cav3.1 T-type channels and HVA currents respectively in INS-1 cells.
| Molecular Weight | 564.57 |
| Formula | C30H38FN3O2.2HCl |
| CAS Number | 357400-13-6 |
| Form | Solid |
| Solubility (25°C) | Water 14.11 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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