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Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.
| Molecular Weight | 367.46 |
| Formula | C18H25NO5S |
| CAS Number | 1138245-21-2 |
| Form | Solid |
| Solubility (25°C) | DMSO 125 mg/mL (ultrasonic) |
| Storage | 4°C, dry, sealed |
[4] J Burgess, et al. Drugs Today (Barc). Mirogabalin besylate in the treatment of neuropathic pain
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