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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M14050 | SCH79797 | SCH79797 is a highly potent, selective nonpeptide protease activated receptor 1 (PAR1) antagonist. |
| M14049 | PAR-4 Agonist Peptide, amide TFA | PAR-4 Agonist Peptide, amide TFA (PAR-4-AP TFA; AY-NH2 TFA) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked by a PAR-4 antagonist. |
| M14048 | GB-88 | GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 µM. |
| M14047 | FSLLRY-NH2 TFA | FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor. |
| M10777 | AGN 194310 | AGN 194310 (VTP-194310) is a highly affinity, potent, selective pan antagonist of retinoic acid receptors (RARs) against RARα, RARβ, RARγ Kd The values are 3 nM, 2 nM, and 5 nM, respectively. |
| M10238 | PAR-2 (6-1) amide (human) | VKGILS-NH2 is a reversed amino acid sequence control peptide for SLIGKV-NH2. |
| M10237 | Protease-Activated Receptor-2, amide | Protease-Activated Receptor-2, amide (SLIGKV-NH2) is a highly potent agonist of PAR2 with IC50 of 10.4 uM. |
| M10236 | PAR-2 (1-6) (mouse, rat) | PAR-2 (1-6) (mouse, rat) is a PAR2 activator, it can be used to explore signaling through PAR2 in cells. |
| M10235 | SLIGRL-NH2 | SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is an agonist of Protease-Activated Receptor-2 (PAR-2). |
| M10143 | AZ3451 | AZ3451 is a potent PAR2 (protease-activated receptor-2) antagonist with IC50 of 23 nM, which plays a part in inflammation response, apoptosis, autophagy and cellular senescence during Osteoarthritis (OA). |
| M9814 | (Ala1)-PAR-4 (1-6) (mouse) | (Ala1)-PAR-4 (1-6) (mouse) |
| M9813 | PAR-4 (1-6) (mouse) | PAR-4 (1-6) (mouse) |
| M9812 | PAR-4 (1-6) (human) | PAR-4 (1-6) (human) is an N-terminal fragment of protease-activated receptor 4 (PAR4) that acts as a PAR4 agonist. |
| M6243 | Vorapaxar Sulfate | Vorapaxar is a first-in-class, potent and orally-active protease-activated receptor 1 (PAR-1) antagonist that blocks thrombin-mediated platelet activation without interfering with thrombin-mediated fibrin deposition. |
| M3123 | Vorapaxar | Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antagonist with Ki of 8.1 nM. |
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