Catalog

PAR Protease-Activated Receptor

Inhibitors

Cat.No.	Name	Information
M10238	PAR-2 (6-1) amide (human)	VKGILS-NH2 is a reversed amino acid sequence control peptide for SLIGKV-NH2.
M10237	Protease-Activated Receptor-2, amide	Protease-Activated Receptor-2, amide (SLIGKV-NH2) is a highly potent agonist of PAR2 with IC50 of 10.4 uM.
M10236	PAR-2 (1-6) (mouse, rat)	PAR-2 (1-6) (mouse, rat) is a PAR2 activator, it can be used to explore signaling through PAR2 in cells.
M10235	SLIGRL-NH2	SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is an agonist of Protease-Activated Receptor-2 (PAR-2).
M10143	AZ3451	AZ3451 is a potent PAR2 (protease-activated receptor-2) antagonist with IC50 of 23 nM, which plays a part in inflammation response, apoptosis, autophagy and cellular senescence during Osteoarthritis (OA).
M9814	(Ala1)-PAR-4 (1-6) (mouse)	(Ala1)-PAR-4 (1-6) (mouse)
M9813	PAR-4 (1-6) (mouse)	PAR-4 (1-6) (mouse)
M9812	PAR-4 (1-6) (human)	PAR-4 (1-6) (human) is an N-terminal fragment of protease-activated receptor 4 (PAR4) that acts as a PAR4 agonist.
M6243	Vorapaxar Sulfate	Vorapaxar is a first-in-class, potent and orally-active protease-activated receptor 1 (PAR-1) antagonist that blocks thrombin-mediated platelet activation without interfering with thrombin-mediated fibrin deposition.
M3123	Vorapaxar	Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antagonist with K_i of 8.1 nM.