Free shipping on all orders over $ 500

FSLLRY-NH2 TFA

Cat. No. M14047
FSLLRY-NH2 TFA Structure
Size Price Availability Quantity
5mg USD 180  USD180 In stock
10mg USD 270  USD270 In stock
25mg USD 480  USD480 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor.

Chemical Information
Molecular Weight 910.98
CAS Number 245329-02-6 (free base)
Solubility (25°C) DMSO 90 mg/mL
Storage -20°C, dry, sealed
Conversion of different model animals based on BSA (PMID: 27057123)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of Compound A used for a mouse (20 mg/kg) to a dose based on the BSA for a rat, multiply 20 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for Compound A of 10 mg/kg.

Related PAR Products
TRAP-6 amide

TRAP-6 amide is a PAR-1 thrombin receptor agonist peptide.

Protease-Activated Receptor-1, PAR-1 Agonist

Protease-Activated Receptor-1, PAR-1 Agonist is a selective proteinase-activated receptor1 (PAR-1) agonist peptide.

FSLLRY-NH2

FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.

iso-TRAP-6

iso-TRAP-6 (iso-SFLLRN) is a PAR-1 agonist that can activate platelets.

PAR-4 Agonist Peptide, amide

PAR-4 Agonist Peptide, amide (PAR-4-AP; AY-NH2) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked by a PAR-4 antagonist.

  Catalog
Abmole Inhibitor Catalog




Keywords: FSLLRY-NH2 TFA supplier, PAR, inhibitors, activators


Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2023 AbMole BioScience. All Rights Reserved.