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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M9911 | IM156 | IM156, a metformin derivative, is an oxidative phosphorylation inhibitor that increases AMPK phosphorylation. |
| M9764 | MK-3903 | MK-3903 is a potent and selective AMPK activator (EC50 = 8 nM). |
| M8095 | PF-06409577 | PF-06409577 is a potent and selective activator of 5′ adenosine monophosphate-activated protein kinase (AMPK). |
| M5336 | Phenformin HCl | Phenformin HCl is a hydrochloride salt of phenformin that is an anti-diabetic drug from the biguanide class. It activates AMPK, increasing activity and phosphorylation. |
| M5326 | HTH-01-015 | HTH-01-015 is a potent and selective NUAK1 inhibitor with IC50 of 100 nM, >100-fold selectivity over NUAK2. |
| M5207 | ETC-1002 | ETC-1002 (ESP-55016) is a novel, first-in-class, orally available, once-daily LDL-C lowering small molecule. |
| M4897 | AICAR | AICAR is an activator of AMP-activated protein kinase (AMPK), down-regulates the insulin receptor expression in HepG2 cells. |
| M4233 | Ginkgolide C | Ginkgolide C is a flavone isolated from Ginkgo biloba leaves, possessing multiple biological functions, such as decreasing platelet aggregation and ameliorating Alzheimer disease. |
| M3946 | BML-275 | BML-275 (Dorsomorphin) is a cell-permeable pyrazolopyrimidine compound shown to be an AMPK inhibitor with Ki of 109 nM in cell-free assays. |
| M3444 | A-769662 | A-769662 is a potent, reversible AMPK activator with EC50of 0.8 μM, little effect on GPPase/FBPase activity. |
| M3244 | Metformin | Metformin is an AMP-activated protein kinase agonist. |
| M3132 | WZ4003 | WZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively, without significant inhibition on 139 other kinases. |
| M2902 | OTSSP167 | OTSSP167 is a highly potent MELK (maternal embryonic leucine zipper kinase) inhibitor with IC50 of 0.41 nM. |
| M2238 | Dorsomorphin (Compound C) dihydrochloride | Dorsomorphin (BML-275) dihydrochloride is a potent inhibitor of AMP-activated protein kinase (AMPK) (Ki = 109 nM) and bone morphogenic protein (BMP) signaling. |
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