Catalog

AhR Aryl Hydrocarbon Receptor

Inhibitors

Cat.No.	Name	Information
M10486	GNF351	GNF351 is a full aryl hydrocarbon receptor (AHR) antagonist. GNF351 competes with a photoaffinity AHR ligand for binding to the AHR with an IC50 of 62 nM.
M10243	D-Kynurenine	D-kynurenine is a metabolite of D-tryptophan, which can be used as a biological precursor of KYNA and 3-hydroxykynurenine.
M9723	L-Kynurenine	L-Kynurenine is an aryl hydrocarbon receptor agonist.
M9714	CAY10465	CAY10465 is an analog of resveratrol acting as a potent and selective aryl hydrocarbon receptor agonist, with a Ki of 0.2 nM.
M9693	PDM2	PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist, with a Ki of 1.2 nM.
M9490	YL-109	YL-109 is a novel anticancer agent, which can inhibit breast cancer cell growth and invasiveness in vitro and in vivo, YL-109 is also an STUB1 enhancer.
M8807	Perillaldehyde	Perillaldehyde inhibits BaP-induced AHR activation and ROS production, inhibits BaP/AHR-mediated release of the CCL2 chemokine, and activats the NRF2/HO1 antioxidant pathway.
M7727	CH-223191	CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist. *The compound is unstable in solutions, freshly prepared is recommended
M4783	Diosimin	Diosimin is a flavonoid glycoside found in citrus fruits, hyssop, and rosemary.
M2577	StemRegenin 1	StemRegenin 1 is an AhR inhibitor with IC50 of 127 nM.