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  Catalog
Abmole Inhibitor Catalog 2017

AChE Acetylcholinesterase

Inhibitors

Cat.No.  Name Information
M8888 Donepezil Donepezil(E 2020) is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM, respectively.
M7585 Atropine Competitive nonselective antagonist at central and peripheral muscarinic acetylcholine receptors.
M6273 Varenicline tartrate Varenicline Tartrate is a nicotinic AChR partial agonist, used to treat nicotine addiction.
M6040 Tropicamide Tropicamide is an anticholinergic and a muscarinic receptor subtype M4-preferring antagonist with IC50 of 8.0 nM.
M5810 Neostigmine methyl sulfate Neostigmine methyl sulfate is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier.
M5604 Edrophonium chloride Edrophonium chloride is a readily reversible acetylcholinesterase inhibitor; prevents breakdown of the neurotransmitter acetylcholine and acts by competitively inhibiting the enzyme acetylcholinesterase, mainly at the neuromuscular junction.
M5433 Atropine Sulfate Monohydrate Atropine sulfate monohydrate is a competitive antagonist for the muscarinic acetylcholine receptor, used to decrease the production of saliva and secretions of the airway prior to surgery.
M5389 Adiphenine Adiphenine HCl is a nicotinic receptor inhibitor with IC50 of 15 μM, used as an antispasmodic drug.
M4188 Tenuifolin Tenuifolin
M3601 Donepezil hydrochloride Donepezil is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM , respectively.
M3590 Butylscopolamine Bromide Butylscopolamine Bromide, is a peripherally acting antimuscarinic, anticholinergic agent used as an abdominal-specific antispasmodic.
M3589 Methscopolamine bromide Methscopolamine is a muscarinic acetylcholine receptor blocker.
M3534 Pancuronium dibromide Pancuronium dibromide is a competitive acetylcholine antagonist with an IC50 of 5.5 nM.
M3453 Scopolamine hydrobromide Scopolamine hydrobromide is a competitive muscarinic acetylcholine receptor with an IC50 of 55.3 nM.
M3309 Bethanechol chloride Bethanechol chloride is a selective muscarinic receptor agonist without any effect on nicotinic receptors.
M3190 PNU-282987 PNU-282987 is a highly selective α7 nAChR agonist with Ki of 27 nM.
M3025 Solifenacin succinate Solifenacin succinate is a urinary antispasmodic of the antimuscarinic class.
M2944 Pilocarpine hydrochloride Pilocarpine hydrochloride is a nonselective muscarinic acetylcholine receptor agonist used to produce an experimental model of epilepsy.
M2762 Hyoscyamine Hyoscyamine is an AChR inhibitor with IC50 of 7.5 nM.
M2613 Darifenacin hydrobromide Darifenacin is a selective M3 muscarinic receptor antagonist with pKi of 8.9.
M2489 Carbachol Carbachol is a cholinomimetic compound that binds and activates the acetylcholine receptor.
M2368 Aclidinium Bromide Aclidinium Bromide inhibits human muscarinic AChR M1, M2, M3, M4 and M5 with Ki of 0.1 nM, 0.14 nM, 0.14 nM, 0.21 nM and 0.16 nM, respectively.
M2268 Rocuronium bromide Rocuronium bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia.


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